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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists
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Reverse Yeast Two-hybrid System to Identify Mammalian Nuclear Receptor Residues that Interact with Ligands and/or Antagonists

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Liver X receptor (LXR) partial agonists: biaryl pyrazoles and imidazoles displaying a preference for LXRβ

Ellen Kick1, Richard Martin2, Yinong Xie2

  • 1Discovery Chemistry, Research & Development, Bristol-Myers Squibb, PO Box 5400, Princeton, NJ 08543-5400, United States.

Bioorganic & Medicinal Chemistry Letters
|December 2, 2014
PubMed

Keywords:
ABCA1LXRLiver X ReceptorNuclear hormone receptorPartial agonist

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