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Characterization at the Molecular Level using Robust Biochemical Approaches of a New Kinase Protein
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Distinct binding mode of multikinase inhibitor lenvatinib revealed by biochemical characterization

Kiyoshi Okamoto1, Megumi Ikemori-Kawada1, Anja Jestel2

  • 1Eisai Co., Ltd , Tsukuba, Ibaraki 300-2635, Japan.

ACS Medicinal Chemistry Letters
|January 16, 2015
PubMed

Keywords:
Receptor tyrosine kinaseVEGFR2X-ray crystallographykinase inhibitorkinetic interaction analysis

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