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Updated: Apr 18, 2026

Using an α-Bungarotoxin Binding Site Tag to Study GABA A Receptor Membrane Localization and Trafficking
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Published on: March 28, 2014

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Regulation of GABAARs by phosphorylation

Yasuko Nakamura1, Laura M Darnieder1, Tarek Z Deeb1

  • 1Department of Neuroscience, Tufts University School of Medicine, Boston, Massachusetts, USA.

Advances in Pharmacology (San Diego, Calif.)
|January 21, 2015
PubMed
Summary

Phosphorylation dynamically regulates gamma-aminobutyric acid type A receptors (GABAARs), impacting their function and expression. Understanding this process is key to addressing neurological disorders linked to GABAAR deficits.

Keywords:
CamKIIGABAGABA(A) receptorInhibitory synapseKinasePKAPKCPhosphatasePhosphorylationSrc

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