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Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers
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Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers

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Enantiomeric cyclic peptides with different Caco-2 permeability suggest carrier-mediated transport

Udaya Kiran Marelli1, Jacqueline Bezençon2, Eduard Puig1

  • 1Institute for Advanced Study and Center for Integrated Protein Science at the Technische Universität München, Department Chemie, Lichtenbergstrasse 4, 85747 Garching (Germany).

Chemistry (Weinheim an Der Bergstrasse, Germany)
|April 29, 2015
PubMed

Keywords:
conformationcyclic peptidesenantioselecitivityintestinal permeabilityoral availability

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