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Biosensor-based affinities and binding kinetics of small molecule antagonists to the adenosine A(2A) receptor

Elena Segala1, James C Errey1, Cédric Fiez-Vandal1

  • 1Heptares Therapeutics, Biopark, Welwyn Garden City, Hertfordshire AL7 3AX, UK.

FEBS Letters
|May 4, 2015
PubMed

Keywords:
G protein-coupled receptorLipid discResidence timeSurface plasmon resonance

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