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Rapid development of two factor IXa inhibitors from hit to lead

Dann L Parker1, Shawn Walsh1, Bing Li1

  • 1Department of Medicinal Chemistry, Merck Research Laboratories, Merck and Co., Inc, PO Box 2000, E. Lincoln Ave., Rahway, NJ 07016, USA.

Bioorganic & Medicinal Chemistry Letters
|May 5, 2015
PubMed

Keywords:
AnticoagulantFactor IXaHit-to-leadParallel synthesisStructure based drug design

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