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Discovery of imidazo[1,5-a]pyridines and -pyrimidines as potent and selective RORc inverse agonists

Benjamin P Fauber1, Alberto Gobbi1, Kirk Robarge1

  • 1Genentech, Inc., 1 DNA Way, South San Francisco, CA 94080, USA.

Bioorganic & Medicinal Chemistry Letters
|June 7, 2015
PubMed

Keywords:
GNE-0946GNE-6468IL-17PPARγRORcRORγ

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