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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Identification and electrophysiological evaluation of 2-methylbenzamide derivatives as Nav1.1 modulators

François Crestey1, Kristen Frederiksen1, Henrik S Jensen1

  • 1§Neuroscience Drug Discovery, H. Lundbeck A/S, Ottiliavej 9, 2500 Valby, Denmark.

ACS Chemical Neuroscience
|June 27, 2015
PubMed

Keywords:
2-Methylbenzamide derivativesNav1.1 modulatorbrain slicesfast-spiking interneuronsvoltage-gated sodium channels

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