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Synthesis and Bioactivity of a Brasilicardin A Analogue Featuring a Simplified Core

Michael E Jung, Brian T Chamberlain, Pierre Koch

  • 1∥NantWorks LLC, Culver City, California 90232, United States.

Organic Letters
|July 7, 2015
PubMed

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Drug design is a dynamic field that involves discovering and developing new medications based on specific biological targets. This process heavily relies on structure-activity relationships (SAR) and quantitative structure-activity relationships (QSAR) to guide the design and optimization of efficient drugs.
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