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Discovery, design, and synthesis of indole-based EZH2 inhibitors

Victor S Gehling1, Rishi G Vaswani1, Christopher G Nasveschuk1

  • 1Constellation Pharmaceuticals, Inc., 215 First Street, Cambridge, MA 02142, USA.

Bioorganic & Medicinal Chemistry Letters
|July 20, 2015
PubMed

Keywords:
EZH2EpigeneticsHistone methyltransferasePRC2Pyridone

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