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Yeast Luminometric and Xenopus Oocyte Electrophysiological Examinations of the Molecular Mechanosensitivity of TRPV4
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Identification of orally-bioavailable antagonists of the TRPV4 ion-channel

Zhi-Liang Wei1, Margaret T Nguyen1, Donogh J R O'Mahony1

  • 1Renovis, Inc. (a wholly-owned subsidiary of Evotec AG), Two Corporate Drive, South San Francisco, CA 94080, United States.

Bioorganic & Medicinal Chemistry Letters
|August 4, 2015
PubMed

Keywords:
AntagonistPainRN-1734RN-9893TRPV4

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