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Structure-Affinity Relationship Analysis of Selective FKBP51 Ligands

Xixi Feng1, Claudia Sippel1, Andreas Bracher2

  • 1Department of Translational Research in Psychiatry, Max Planck Institute of Psychiatry , Kraepelinstrasse 2, 80804 Munich, Germany.

Journal of Medicinal Chemistry
|October 1, 2015
PubMed
Summary

Researchers developed novel, smaller selective ligands for FKBP51, a key target for psychiatric and metabolic disorders. These compounds bind to FKBP51

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