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Updated: Mar 30, 2026

Synthesis of 1,2-Azaborines and the Preparation of Their Protein Complexes with T4 Lysozyme Mutants
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Benzazaborinines as Novel Bioisosteric Replacements of Naphthalene: Propranolol as an Example

Frederik J R Rombouts1, Fulgencio Tovar2, Nigel Austin3

  • 1Neuroscience-Medicinal Chemistry, Janssen Research & Development, Janssen Pharmaceutica N.V. , Turnhoutseweg 30, B-2340 Beerse, Belgium.

Journal of Medicinal Chemistry
|November 14, 2015
PubMed

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