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Flat SAR of P3-methylsulphonamide based small molecule legumain inhibitors

Kerry Anne Ness1, Sharon L Eddie1, Stephanie Burton2

  • 1CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, UK.

Bioorganic & Medicinal Chemistry Letters
|December 15, 2015
PubMed

Keywords:
CancerLegumainSARSmall molecule protease inhibitor

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