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Symmetric 4,4'-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulators

Manabu Sato1, Kiminori Ohta1, Asako Kaise1

  • 1Faculty of Pharmaceutical Sciences, Tohoku Pharmaceutical University, 4-4-1 Komatsushima, Aoba-ku, Sendai 981-8558, Japan.

Bioorganic & Medicinal Chemistry
|January 30, 2016
PubMed

Keywords:
2,2,6,6-TetramethylpiperidineEstrogen receptor modulatorHydrophobicityMcMurry couplingPiperidine

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