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Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of sulphone-based CRTh2 antagonists

Maria Antonia Buil1, Marta Calbet1, Marcos Castillo2

  • 1Almirall R&D Centre, Laureano Miró, 408-410, 08980, Sant Feliu de Llobregat, Barcelona, Spain.

European Journal of Medicinal Chemistry
|February 29, 2016
PubMed

Keywords:
CRTh2 antagonistReceptor residence timeStructure-activity relationship (SAR)Structure-kinetic relationship (SKR)

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