Related Experiment Video

Updated: Jul 26, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
07:16

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

[EXPERIMENTAL PHARMACOKINETICS AND PHARMACODYNAMICS OF GB-115 DIPEPTIDE ANXIOLYTIC SUBSTANCES].

L G Kolik, V P Zherdev, S S Boiko

    Eksperimental'Naia I Klinicheskaia Farmakologiia
    |March 29, 2016
    PubMed
    Summary

    Micronized GB-115, a dipeptide anxiolytic, shows improved pharmacokinetics and bioavailability in rats compared to its crystalline form. The micronized substance also demonstrated superior anxiolytic effects in the elevated plus maze test.

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