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New P2X3 receptor antagonists. Part 1: Discovery and optimization of tricyclic compounds

Gábor Szántó1, Attila Makó1, Imre Bata1

  • 1Gedeon Richter Plc, Budapest 10, PO Box 27, H-1475, Hungary.

Bioorganic & Medicinal Chemistry Letters
|July 18, 2016
PubMed

Keywords:
ATPAirway hyperractivityChiralityHTS campaignIon channelNew binding siteP2X3 antagonistPurinergic receptor

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