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Optimization of microtubule affinity regulating kinase (MARK) inhibitors with improved physical properties

David L Sloman1, Njamkou Noucti1, Michael D Altman2

  • 1Discovery Chemistry, Merck and Co., Inc., 33 Avenue Louis Pasteur, Boston, MA 02215, United States.

Bioorganic & Medicinal Chemistry Letters
|August 6, 2016
PubMed

Keywords:
Alzheimer’s diseaseAmine basicityFluorineKinaseMARK

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