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Updated: Mar 13, 2026

A High-throughput-compatible FRET-based Platform for Identification and Characterization of Botulinum Neurotoxin Light Chain Modulators
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Picolinic acids as β-exosite inhibitors of botulinum neurotoxin A light chain

Paul T Bremer1, Song Xue1, Kim D Janda1

  • 1Departments of Chemistry, Immunology and Microbial Sciences, Worm Institute for Research and Medicine (WIRM), The Scripps Research Institute, 10550 N. Torrey Pines Rd, La Jolla, CA 92037, USA. kdjanda@scripps.edu.

Chemical Communications (Cambridge, England)
|October 11, 2016
PubMed

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