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Updated: Mar 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Discovery and Characterization of Novel GPR39 Agonists Allosterically Modulated by Zinc

Seiji Sato1, Xi-Ping Huang1, Wesley K Kroeze1

  • 1Department of Pharmacology (S.S., X.-P.H., W.K.K., B.L.R.) and National Institute of Mental Health Psychoactive Drug Screening Program (X.-P.H., B.L.R.), School of Medicine, University of North Carolina, Chapel Hill, North Carolina.

Molecular Pharmacology
|November 3, 2016
PubMed

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