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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists

Gilles Ouvry1, Claire Bouix-Peter1, Fabrice Ciesielski2

  • 1Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.

Bioorganic & Medicinal Chemistry Letters
|November 6, 2016
PubMed

Keywords:
AllostericInverse agonistsPhototoxicityROR gammaTopical administration

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