Designed covalent allosteric modulators: an emerging paradigm in drug discovery

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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Shaoyong Lu1, Jian Zhang2

  • 1Department of Pathophysiology, Shanghai Key Laboratory of Tumor Microenvironment and Inflammation, Key Laboratory of Cell Differentiation and Apoptosis of Chinese Ministry of Education, Shanghai Jiao Tong University, School of Medicine, Shanghai 200025, China.

Drug Discovery Today
|November 27, 2016
PubMed

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