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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Identification of an Orally Efficacious GPR40/FFAR1 Receptor Agonist

Sameer Agarwal1, Santosh Sasane1, Prashant Deshmukh1

  • 1Zydus Research Centre, Cadila Healthcare Ltd. , Sarkhej-Bavla N.H. No. 8 A, Moraiya, Ahmedabad-382 210, India.

ACS Medicinal Chemistry Letters
|December 21, 2016
PubMed

Keywords:
FFAR1GPR40GPR40 agonistfatty acidsinsulin secretiontype 2 diabetes

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