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Updated: Jun 27, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

Structure-Based Design of Highly Selective Inhibitors of the CREB Binding Protein Bromodomain

R Aldrin Denny1, Andrew C Flick2, Jotham Coe2

  • 1Medicine Design, Pfizer , 610 Main Street, Cambridge Massachusetts 02139, United States.

Journal of Medicinal Chemistry
|April 5, 2017
PubMed

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