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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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A multifunctional catalyst that stereoselectively assembles prodrugs

Daniel A DiRocco1, Yining Ji2, Edward C Sherer2

  • 1Process Research and Development, Merck & Co., Inc., Rahway, NJ 07065, USA. daniel.dirocco@merck.com.

Science (New York, N.Y.)
|April 29, 2017
PubMed

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