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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Discovery of a highly potent, selective and novel CDK9 inhibitor as an anticancer drug candidate

Yongtao Li1, Qingxiang Guo1, Chao Zhang2

  • 1School of Medicine, Nankai University, 94 Weijin Road, Tianjin 300071, China; Tianjin International S & T Cooperation Base, 94 Weijin Road, Tianjin 300071, China.

Bioorganic & Medicinal Chemistry Letters
|June 28, 2017
PubMed

Keywords:
CDK9CancerInhibitorLEE011

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