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Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles

Martin Hügle1, Xavier Lucas2, Dmytro Ostrovskyi3

  • 1Institut für Biochemie, Albert-Ludwigs-Universität Freiburg, Albertstrasse 21, 79104, Freiburg, Germany.

Angewandte Chemie (International Ed. in English)
|August 3, 2017
PubMed

Keywords:
4-acyl pyrrolesCBPbromodomainsdrug discoveryp300

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