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Identification of potent lysophosphatidic acid receptor 5 (LPA5) antagonists as potential analgesic agents

Yuichiro Kawamoto1, Ryushi Seo1, Nobuhito Murai1

  • 1Drug Discovery Research, Astellas Pharma Inc., 21 Miyukigaoka, Tsukuba, Ibaraki 305-8585, Japan.

Bioorganic & Medicinal Chemistry
|December 7, 2017
PubMed

Keywords:
Analgesic agentsBBB permeabilityCNS MPO scoreHomology modelLPA5 antagonist

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