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Updated: Feb 17, 2026

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Transactivation Assays that Identify Indirect and Direct Activators of Human Pregnane X Receptor (PXR, NR1I2) and

Marija Pinne1, Elsa Ponce1, Judy L Raucy1

  • 1Puracyp, Inc., Carlsbad, CA 92010, United States.

Drug Metabolism Letters
|December 9, 2017
PubMed
Abstract

Keywords:
CARDPX2 cellsLigand binding assaysPXRdrug-drug interactionsfull length nuclear receptorindirect activatorsnuclear receptorsphenobarbitalphosphorylation

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