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Antineoplastic Agents. 606. The Betulastatins

George R Pettit1, Noeleen Melody1, Jean-Charles Chapuis1

  • 1Department of Chemistry and Biochemistry , Arizona State University , P.O. Box 871604, Tempe , Arizona 85287-1604 , United States.

Journal of Natural Products
|January 6, 2018
PubMed
Summary

Researchers modified betulin, a plant compound, to create novel anticancer agents called betulastatins. Betulastatin 3 demonstrated significant cancer cell growth inhibition, showing promise for further drug development.

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