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Structure-activity relationships of HDAC8 inhibitors: Non-hydroxamates as anticancer agents

Sk Abdul Amin1, Nilanjan Adhikari1, Tarun Jha1

  • 1Natural Science Laboratory, Division of Medicinal and Pharmaceutical Chemistry, Department of Pharmaceutical Technology, P. O. Box 17020, Jadavpur University, Kolkata, 700032, West Bengal, India.

Pharmacological Research
|March 8, 2018
PubMed

Keywords:
CancerHDAC8 inhibitorHistone deacetylaseNon-hydroxamatesPCI-34051 (PubChem CID: 24753719)Romidepsin (PubChem CID: 5352062)Structure-activity relationship (SAR)Vorinostat (PubChem CID: 5311)Zinc binding group

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