Virtual Fragment Screening Identification of a Quinoline-5,8-dicarboxylic Acid Derivative as a Selective JMJD3

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Assunta Giordano1,2, Federica Del Gaudio2,3,4, Catrine Johansson5

  • 1Institute of Biomolecular Chemistry (ICB), Consiglio Nazionale delle Ricerche (CNR), Via Campi Flegrei 34, 80078, Pozzuoli (Napoli), Italy.

Chemmedchem
|April 11, 2018
PubMed

Keywords:
anticancer agentsdrug discoveryfragment-based approachmolecular modelingselective JMJD3 inhibitor

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