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PF-06827443 Displays Robust Allosteric Agonist and Positive Allosteric Modulator Activity in High Receptor Reserve

Sean P Moran1,2,3, Hyekyung P Cho2,3, James Maksymetz2,3

  • 1Vanderbilt Brain Institute , Vanderbilt University , Nashville , Tennessee 37232 , United States.

ACS Chemical Neuroscience
|April 24, 2018
PubMed

Keywords:
Alzheimer’s diseaseM1Positive allosteric modulatorago-PAMlong-term depressionmuscarinic acetylcholine receptorprefrontal cortexschizophrenia

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