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PAM-Antagonists: A Better Way to Block Pathological Receptor Signaling?

Terry Kenakin1, Ryan T Strachan1

  • 1Department of Pharmacology, University of North Carolina School of Medicine, Chapel Hill, NC, USA.

Trends in Pharmacological Sciences
|June 11, 2018
PubMed

Keywords:
drug discoverynegative allosteric modulationreceptor antagonismreceptor theoryselective drug antagonism

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