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Discovery and hit-to-lead evaluation of piperazine amides as selective, state-dependent NaV1.7 inhibitors

Brian A Sparling1, S Yi1, J Able2

  • 1Department of Medicinal Chemistry , Amgen Inc. , 360 Binney Street , Cambridge , MA 02142 , USA .

Medchemcomm
|August 16, 2018
PubMed

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