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Design, synthesis, and discovery of ocotillol-type amide derivatives as orally available modulators of

Qianwen Ren1, Gangqiang Yang1, Mengqi Guo2

  • 1School of Pharmacy, Collaborative Innovation Center of Advanced Drug Delivery System and Biotech Drugs in Universities of Shandong, Key Laboratory of Molecular Pharmacology and Drug Evaluation (Yantai University), Ministry of Education, Yantai University, Yantai, 264005, China.

European Journal of Medicinal Chemistry
|October 23, 2018
PubMed

Keywords:
Molecular dockingMultidrug resistance reversalOcotillolP-glycoprotein modulatorsStructure-active relationship

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