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Updated: Jan 31, 2026

Quantifying Agonist Activity at G Protein-coupled Receptors
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Quantifying Agonist Activity at G Protein-coupled Receptors

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Dual conformation of the ligand induces the partial agonistic activity of retinoid X receptor α (RXRα)

Yurina Miyashita1,2,3, Nobutaka Numoto3, Sundaram Arulmozhiraja1,4

  • 1Department of Chemistry, Rikkyo University, Tokyo, Japan.

FEBS Letters
|December 20, 2018
PubMed

Keywords:
RXRαbiochemical analysiscrystal structurefragment molecular orbital theorymolecular dynamics simulationspartial agonist

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