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Synthesis and evaluation of haloperidol ester prodrugs metabolically activated by human carboxylesterase

Masato Takahashi1, Tomoki Uehara1, Minori Nonaka1

  • 1Faculty of Pharmacy, Chiba Institute of Science, 15-8, Shiomi-cho, Choshi, Chiba 288-0025, Japan.

European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences
|March 18, 2019
PubMed

Keywords:
CarboxylesteraseEnol esterHaloperidolProdrugSustained release

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