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Benzothiophene derivatives as phosphodiesterase 10A (PDE10A) inhibitors: Hit-to-lead studies

Yoshito Kawamoto1, Minako Tomino1, Kenichi Hiramatsu1

  • 1Asubio Pharma Co., Ltd., 6-4-3 Minatojima-Minamimachi, Chuo-ku, Kobe, Hyogo 650-0047, Japan.

Bioorganic & Medicinal Chemistry Letters
|April 7, 2019
PubMed

Keywords:
BenzothiopheneConformational alterationHit-to-lead studiesPDE10A inhibitorsPhosphodiesterase 10A inhibitors

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