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1-Phenyl-dihydrobenzoindazoles as novel colchicine site inhibitors: Structural basis and antitumor efficacy

Junhang Jiang1, Hao Zhang2, Chongqing Wang1

  • 1School of Pharmacy, Second Military Medical University, 325 Guohe Road, Shanghai, 200433, China.

European Journal of Medicinal Chemistry
|June 8, 2019
PubMed

Keywords:
Cis-trans photoisomerizationColchicine site inhibitorsMicrotubule-targeting agentsWater-soluble prodrugX-ray co-crystal structure

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