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Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflow

Xavier Fradera1, Joey L Methot2, Abdelghani Achab2

  • 1Computational and Structural Chemistry, Merck & Co., Inc., Boston, MA, USA.

Bioorganic & Medicinal Chemistry Letters
|August 17, 2019
PubMed

Keywords:
OxindolePI3KδScaffold-hoppingStructure-based drug design

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