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Updated: Jan 19, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors

Ann L Walker1, Alexis Denis1, Ryan P Bingham1

  • 1GlaxoSmithKline R&D, Medicines Research Centre, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, UK.

Bioorganic & Medicinal Chemistry Letters
|September 16, 2019
PubMed

Keywords:
KLK1KLK5KLKB1LEKTINetherton syndromeSPINK5

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