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Updated: Dec 31, 2025

A "Dual-Addition" Calcium Fluorescence Assay for the High-Throughput Screening of Recombinant G Protein-Coupled Receptors
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Identification of novel GPR81 agonist lead series for target biology evaluation

Öjvind Davidsson1, Kristina Nilsson1, Jonas Brånalt1

  • 1CVRM Medicinal Chemistry, Research and Early Development, Cardiovascular, Renal and Metabolism, BioPharmaceuticals R&D, AstraZeneca, Gothenburg, Sweden.

Bioorganic & Medicinal Chemistry Letters
|January 15, 2020
PubMed

Keywords:
GHSR1aGPCRGPR109AGPR81HTSLipolysis

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