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Focused structure-activity relationship profiling around the 2-phenylindole scaffold of a cannabinoid type-1 receptor

Peter C Schaffer1, Pushkar M Kulkarni1, David R Janero2

  • 1Department of Pharmaceutical Sciences, Bouvé College of Health Sciences, Northeastern University, Boston, MA 02115, United States.

Bioorganic & Medicinal Chemistry
|October 16, 2020
PubMed

Keywords:
2-PhenylindoleCannabinoid type-1 receptorFunctional selectivityPhysiochemical propertiesPositive allosteric modulator

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