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Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK

Anurag S Srivastava1, Soo Ko1, Scott H Watterson1

  • 1Bristol Myers Squibb Research and Early Development, P.O. Box 4000, Princeton, New Jersey 08543, United States.

ACS Medicinal Chemistry Letters
|November 20, 2020
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