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Sublingual Estradiol Is Associated with Higher Estrone Concentrations than Transdermal or Injectable Preparations in

Lauren R Cirrincione1, Gabrielle Winston McPherson2, Jessica Rongitsch3

  • 1Department of Pharmacy, University of Washington, Seattle, Washington, USA.

LGBT Health
|January 13, 2021
PubMed
Summary

Serum estrone levels were higher with sublingual estradiol compared to transdermal or injectable forms in feminizing gender-affirming hormone therapy (GAHT). Estradiol levels varied by injection versus transdermal methods but not with sublingual use.

Keywords:
estradiolestronegender-affirming hormone therapytransgendertransgender women

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