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Updated: Nov 19, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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The Three-Component Synthesis of 4-Sulfonyl-1,2,3-triazoles via a Sequential Aerobic Copper-Catalyzed Sulfonylation

Max Van Hoof1, Santhini Pulikkal Veettil1, Wim Dehaen1

  • 1Molecular Design and Synthesis, Department of Chemistry, KU Leuven, 3001 Leuven, Belgium.

Molecules (Basel, Switzerland)
|January 27, 2021
PubMed

Keywords:
4-sulfonyl-1,2,3-triazolesC-H activationDimroth azide–enolate cyclizationaerobic oxidationcopper-catalysisthree-component tandem reaction

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