Genetic Polymorphism Effect on Warfarin-Rifampin Interaction: A Case Report and Review of Literature

Muhammad Salem1, Islam Eljilany2, Ahmed El-Bardissy1

  • 1Department of Pharmacy, Hamad General Hospital, Doha, Qatar.

Insights

Genetic factors influence warfarin dosing during rifampin treatment. A patient with specific gene variants achieved therapeutic international normalized ratio (INR) levels on a lower warfarin dose, suggesting genotype impacts this drug interaction.

Area of Science:

  • Pharmacogenomics
  • Drug Interactions
  • Internal Medicine

Background:

  • The interaction between warfarin and rifampin is well-documented, with rifampin's induction of CYP2C9 often necessitating high warfarin doses.
  • Genetic polymorphisms in warfarin-metabolizing enzymes and targets significantly affect individual dose requirements, accounting for up to 50% of variability.

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