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Exploring the putative mechanism of allosteric modulations by mixed-action kappa/mu opioid receptor bitopic

Huiqun Wang1, Danni Cao2, James C Gillespie3

  • 1Department of Medicinal Chemistry, School of Pharmacy, Virginia Commonwealth University, Richmond, VA 23298, USA.

Future Medicinal Chemistry
|February 16, 2021
PubMed

Keywords:
allosteric modulation mechanismkappa opioid receptor (KOR)/mu opioid receptor (MOR)mixed-action KOR/MOR ligandmolecular dynamics simulationspsychostimulant abuse and addictionselectivity

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